Circumventing seizure activity in a series of G Protein Coupled Receptor 119 (GPR119) agonists
Bradley Shaw2017-11-07T13:51:35+00:00100) Circumventing seizure activity in a series of G Protein Coupled Receptor 119 (GPR119)
Medicinal chemistry optimisation of kinetics” in Kinetics and Thermodynamics of Drug Binding
Bradley Shaw2017-11-07T13:50:58+00:00101) Medicinal chemistry optimisation of kinetics” in Kinetics and Thermodynamics of Drug Binding, Keseru,
Tactics to avoid inhibition of cytochrome P450s” in Tactics in Contemporary Drug Design
Bradley Shaw2017-11-07T13:50:32+00:00101) Tactics to avoid inhibition of cytochrome P450s” in Tactics in Contemporary Drug Design,
Discovery of a series of 2-(pyridinyl)pyrimidines as potent antagonists of GPR40.
Bradley Shaw2017-11-07T13:50:01+00:00102) Discovery of a series of 2-(pyridinyl)pyrimidines as potent antagonists of GPR40. Waring, M.
An Orally Bioavailable, Indole-3-glyoxylamide Based Series of Tubulin Polymerization Inhibitors Showing Tumor Growth Inhibition in a Mouse Xenograft Model of Head and Neck Cancer.
Bradley Shaw2017-11-07T13:49:20+00:00103) An Orally Bioavailable, Indole-3-glyoxylamide Based Series of Tubulin Polymerization Inhibitors Showing Tumor Growth
A mechanistic proposal for the protodeboronation of neat boronic acids: boronic acid mediated reaction in the solid state.
Bradley Shaw2017-11-07T13:48:44+00:00104) A mechanistic proposal for the protodeboronation of neat boronic acids: boronic acid mediated
Designing hydroxamates and reversed hydroxamates to inhibit zinc-containing proteases but not cytochrome P450s: insights from quantum mechanics and protein-ligand crystal structures
Bradley Shaw2017-11-07T13:04:03+00:00105) Designing hydroxamates and reversed hydroxamates to inhibit zinc-containing proteases but not cytochrome P450s:
Novel N-thiazolyl piperazine-1-carboxamide CCR2 antagonists – investigation of an unexpected reaction with glutathione
Bradley Shaw2017-11-07T13:03:20+00:00106) Novel N-thiazolyl piperazine-1-carboxamide CCR2 antagonists – investigation of an unexpected reaction with glutathione.
Protodeboronation of Heteroaromatic, Vinyl, and Cyclopropyl Boronic Acids: pH-Rate Profiles, Autocatalysis, and Disproportionation.
Bradley Shaw2017-11-07T13:02:28+00:00Protodeboronation of Heteroaromatic, Vinyl, and Cyclopropyl Boronic Acids: pH-Rate Profiles, Autocatalysis, and Disproportionation. Cox,
“Matched molecular pair analysis” in Comprehensive Medicinal Chemistry III
Bradley Shaw2017-11-07T13:01:28+00:00109) “Matched molecular pair analysis” in Comprehensive Medicinal Chemistry III, Davis, A. and Edge,
