Achieving improved permeability by hydrogen bond donor modulation in a series of MGAT2 inhibitors.

2017-11-07T13:57:54+00:00

94) Achieving improved permeability by hydrogen bond donor modulation in a series of MGAT2 inhibitors. Scott. J. S.; Berry, D. J.; Brown, H. S.; Buckett, L.; Clarke, D. S.; Goldberg, K.; Hudson, J. A.; Leach, A. G.; MacFaul, P. A.; Raubo, P.; Robb, G. R. Med. Chem. Comm. 2013, 4, 1305-1311.

Achieving improved permeability by hydrogen bond donor modulation in a series of MGAT2 inhibitors.2017-11-07T13:57:54+00:00

Optimization of Brain Penetrant 11β-Hydroxysteroid Dehydrogenase Type I Inhibitors and in Vivo Testing in Diet-Induced Obese Mice

2017-11-07T13:56:13+00:00

96) Optimization of Brain Penetrant 11β-Hydroxysteroid Dehydrogenase Type I Inhibitors and in Vivo Testing in Diet-Induced Obese Mice Goldberg, F.W.; Dossetter, A.G.; Scott, J.S. Robb, G.R; Boyd, S.; Groombridge, S.D.; Kemmitt, P.D.; Sjogren, T.; Morentin-Gutierrez, P.; deSchoolmeester, J.; Swales, J.G.; Turnbull, A.V.; Wild, M.J. J. Med. Chem. 2014,57 (3), pp 970-986. DOI: 10.1021/jm4016729

Optimization of Brain Penetrant 11β-Hydroxysteroid Dehydrogenase Type I Inhibitors and in Vivo Testing in Diet-Induced Obese Mice2017-11-07T13:56:13+00:00

Identification, Optimization, and Pharmacology of Acylurea GHS-R1a Inverse Agonists

2017-11-07T13:55:32+00:00

97) Identification, Optimization, and Pharmacology of Acylurea GHS-R1a Inverse Agonists McCoull, W.; Barton, P., Brown, A. J. H. ; Bowker, S.S.; Cameron, J.; Clarke, D.S.; Davies, R. D. M.; Dossetter, A.G.; Ertan, A.; Fenwick, M.; Green, C.; Holmes, J.L.; Martin, N.; Masters, D.; Moore, J.E.; Newcombe, N.J.; Newton, C.; Pointon, H.; Robb, G.R.; Sheldon, C.;

Identification, Optimization, and Pharmacology of Acylurea GHS-R1a Inverse Agonists2017-11-07T13:55:32+00:00

Circumventing seizure activity in a series of G Protein Coupled Receptor 119 (GPR119) agonists

2017-11-07T13:51:35+00:00

100) Circumventing seizure activity in a series of G Protein Coupled Receptor 119 (GPR119) agonists. Scott, J. S.; Bowker, S. S.; Brocklehurst, K. J.; Brown, H. S.; Clarke, D. S.; Easter, A.; Ertan, A.; Goldberg, K. Hudson, J. A.; Kavanagh, S.; Laber, D.; Leach, A. G.; MacFaul, P. A.; Martin, E. A.; McKerrecher, D.; Schofield,

Circumventing seizure activity in a series of G Protein Coupled Receptor 119 (GPR119) agonists2017-11-07T13:51:35+00:00
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