81) Identification of pyrazolo-pyrimidinones as GHS-R1a antagonists and inverse agonists for the treatment of obesity. McCoull W, Barton P, Broo A, Brown A, Clarke D, Coope G, Davies RDM, Dossetter AG , Kelly E,  Knerr L, Macfaul P, Holmes J,  Martin N,  Moore JE, Morgan D, Newton C, Osterlund K, Robb G, Rosevere E, Selmi N, Stokes S, Svensson T, Ullah V, Williams, E. Med. Chem. Commun., 2012, Accepted Manuscript