61) Quantitatively Interpreted Enhanced Inhibition of Cytochrome P450s by Heteroaromatic Rings Containing Nitrogen Leach, A. G.*; Kidley, N. J. J. Chem. Inf. Model. 2011, 51, 1048-1063.

62) “The Discovery of Benzanilides as c-Met Receptor Tyrosine Kinase Inhibitors by a Directed Screening approach” Allen, J. V.; Bardelle, C.; Blades, K.; Buttar, D.; Chapman, L.; Colclough, N.; Dossetter, A. G.; Garner, A. P.; Girdwood, A.; Lambert, C.; Leach, A. G.; Law, B.; Major, J.; Plant, H.; Slater, A. M. Bioorganic & Medicinal Chemistry

63) Matched Molecular Pairs as a Medicinal Chemistry Tool Griffen, E.; Leach, A. G.*; Robb, G. R.; Warner, D. J. J. Med. Chem. 2011, 54, 7739-7750.

64) “Discovery, optimisation and in vivo evaluation of novel GPR119 agonists” Brocklehurst, K. J.; Broo, A.; Butlin, R. J.; Brown, H. S.; Clarke, D. S.; Davidsson, Ö.; Goldberg, K.; Groombridge, S. D.; Kelly, E. E.; Leach, A.; McKerrecher, D.; O’Donnell, C.; Poucher, S.; Schofield, P.; Scott, J. S.; Teague, J.; Westgate, L.; Wood, M. J.

65) DNA-dependent protein kinase (DNA-PK) inhibitors: Structure-activity relationships for O-alkoxyphenylchromen-4-one probes of the ATP-binding domain Clapham, Kate M.; Bardos, Julia; Finlay, M. Raymond V.; Golding, Bernard T.; Griffen, Edward J.; Griffin, Roger J.; Hardcastle, Ian R.; Menear, Keith A.; Ting, Attilla; Turner, Paul;  et al  Bioorganic & Medicinal Chemistry Letters (2011), 21(3), 966-970.DOI: 10.1016/j.bmcl.2010.12.047

66) “Do Glycosyl Sulfonium Ions Engage in Neighbouring-Group Participation? A Study of Oxathiane Glycosyl Donors and the Basis for their Stereoselectivity” Fascione, M. A.; Kilner, C. A.; Leach, A. G.; Turnbull, W. B. Chem. Eur. J. 2012, 18, 321-333.

67) “Mechanistic Studies on a Sulfoxide Transfer Reaction Mediated by Diphenyl Sulfoxide/Triflic Anhydride” Fascione, M. A.; Adshead, S. J.; Mandal, P. K.; Kilner, C. A.; Leach, A. G.; Turnbull, W. B. Chem. Eur. J. 2012, 18, 2987-2997.

68) Enantiomeric pairs reveal that key medicinal chemistry parameters vary more than simple physical property based models can explain Andrew G. Leach, Elizabeth A. Pilling, Alfred A. Rabow, Simone Tomasi, Nabil Asaad, Niklaas J. Buurma, Andrew Ballard and Stefania Narduolo Med. Chem. Commun., 2012,3, 528-540.

69) Oxadiazole isomers: all bioisosteres are not created equal Kristin Goldberg, Sam Groombridge, Julian Hudson, Andrew G. Leach, Philip A. MacFaul, Adrian Pickup, Ruth Poultney, James S. Scott, Per H. Svensson and Joseph Sweeney Med. Chem. Commun., 2012,3, 600-604.

70) Rationally Designing Safer Anilines: The Challenging Case of 4-Aminobiphenyls Birch, A. M.; Groombridge, S.; Law, R.; Leach, A. G.*; Mee, C.; Schramm, C. J. Med. Chem. 2012, 55, 3923-3933.